Tolinapant (ASTX-660)
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | ASTX660 is an orally bioavailable, non-peptidomimetic antagonist of both X chromosome-linked inhibitor of apoptosis protein (XIAP) and cellular IAP 1 (cIAP1), with potential antineoplastic and pro-apoptoticctivities. 1799328-86-1 (free base) 1799328-50-9 (HCl) 1799328-90-7 (mesylate) 1799328-88-3 (sulfate) |
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Catalog Num | A16996 |
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Formula | C30H42FN5O3 |
Molecular Weight | 539.69 |
CAS Number | 1799328-86-1 |
SMILES | OCC1=NC2=C(N(CC2(C)C)C(CN3[C@@H](CN4[C@H](C)COCC4)CN[C@H](C)C3)=O)C=C1CC5=CC=C(F)C=C5 |
Synonyms | ASTX660, ASTX 660 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 93 mg/mL (172.32 mM) | |
Water | Insoluble | ||
Ethanol | 93 mg/mL (172.32 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 18.53 mL | 92.65 mL | 185.29 mL |
0.5 mM | 3.71 mL | 18.53 mL | 37.06 mL |
1 mM | 1.85 mL | 9.26 mL | 18.53 mL |
5 mM | 0.37 mL | 1.85 mL | 3.71 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2