GSK6853

Name: GSK6853
SKU: A16330
Price: 80 USD
Rating: 5 (288 reviews)

Catalog No.: A16330

BRPF1 bromodomain inhibitor

GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. shows excellent BRPF1 potency (pKd 9.5) and greater than 1600-fold selectivity over all other bromodomains tested.

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Data Sheet

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Biological Activity

Discription	GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. shows excellent BRPF1 potency (pKd 9.5) and greater than 1600-fold selectivity over all other bromodomains tested.

Product Information

Catalog Num	A16330
Formula	C22H27N5O3
Molecular Weight	409.48
CAS Number	1910124-24-1
SMILES	O=C(NC1=C(N2[C@H](C)CNCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC
Synonyms	GSK-6853, GSK 6853
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro	DMSO	Warmed: 77 mg/mL (188.04 mM)
	Water	Insoluble
	Ethanol	Warmed: 77 mg/mL (188.04 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	24.42 mL	122.11 mL	244.21 mL
0.5 mM	4.88 mL	24.42 mL	48.84 mL
1 mM	2.44 mL	12.21 mL	24.42 mL
5 mM	0.49 mL	2.44 mL	4.88 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Product Name	Price	Stock
GSK6853 5mg	$80.00	In stock
GSK6853 10mg	$140.00	In stock
GSK6853 50mg	$420.00	In stock
Bulk Size	Bulk Discount