Relugolix

Catalog No.: A17783
GnRH antagonist
Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013.
Grouped product items
Product Name Price Stock Qty
Relugolix 1mg
$60.00
In stock
Relugolix 5mg
$110.00
In stock
Relugolix 10mg
$180.00
In stock
Relugolix 50mg
$600.00
In stock
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Important Notice: For research use only. We do not sell to patients.

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Biological Activity
Discription Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013.
Product Information
Catalog Num A17783
Formula C29H27F2N7O5S
Molecular Weight 623.63
CAS Number 737789-87-6
SMILES O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)C)C(C(N3C4=NN=C(OC)C=C4)=O)=C2N(CC5=C(F)C=CC=C5F)C3=O)C=C1
Synonyms TAK385; TAK-385; TAK 385; Relugolix.
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 59 mg/mL (94.6 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.04 mL 80.18 mL 160.35 mL
0.5 mM 3.21 mL 16.04 mL 32.07 mL
1 mM 1.6 mL 8.02 mL 16.04 mL
5 mM 0.32 mL 1.6 mL 3.21 mL
Useful Calculator

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