Relugolix
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. |
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Catalog Num | A17783 |
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Formula | C29H27F2N7O5S |
Molecular Weight | 623.63 |
CAS Number | 737789-87-6 |
SMILES | O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)C)C(C(N3C4=NN=C(OC)C=C4)=O)=C2N(CC5=C(F)C=CC=C5F)C3=O)C=C1 |
Synonyms | TAK385; TAK-385; TAK 385; Relugolix. |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 59 mg/mL (94.6 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 16.04 mL | 80.18 mL | 160.35 mL |
0.5 mM | 3.21 mL | 16.04 mL | 32.07 mL |
1 mM | 1.6 mL | 8.02 mL | 16.04 mL |
5 mM | 0.32 mL | 1.6 mL | 3.21 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2