ICEC0942 HCl

Catalog No.: A16903
CDK7 inhibitor
ICEC0942, also known as CT7001, is an Orally Bioavailable Selective Inhibitor of CDK7 for Cancer Treatment. It selectively inhibits CDK7, with an IC50 of 40nM; IC50 values for CDK1, CDK2, CDK5 and CDK9 were 45-, 15-, 230- and 30-fold higher.
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Product Name Stock
ICEC0942 HCl 5mg
ICEC0942 HCl 10mg
ICEC0942 HCl 50mg
ICEC0942 HCl 100mg
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Biological Activity
Discription ICEC0942, also known as CT7001, is an Orally Bioavailable Selective Inhibitor of CDK7 for Cancer Treatment. It selectively inhibits CDK7, with an IC50 of 40nM; IC50 values for CDK1, CDK2, CDK5 and CDK9 were 45-, 15-, 230- and 30-fold higher.
Targets
Target Value
Product Information
Catalog Num A16903
Formula C22H31ClN6O
Molecular Weight 430.98
CAS Number 1805789-54-1
SMILES O[C@H]1CNCC[C@@H]1CNC2=NC3=C(C(C)C)C=NN3C(NCC4=CC=CC=C4)=C2.[H]Cl
Synonyms CT7001
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 76 mg/mL (176.34 mM)
Water 76 mg/mL (176.34 mM)
Ethanol 13 mg/mL (30.16 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.2 mL 116.01 mL 232.03 mL
0.5 mM 4.64 mL 23.2 mL 46.41 mL
1 mM 2.32 mL 11.6 mL 23.2 mL
5 mM 0.46 mL 2.32 mL 4.64 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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