PF-06821497

Catalog No.: A21388
EZH2 inhibitor
PF-06821497 (compound 23a) is a potent, selective and orally active Enhancer of Zeste Homolog 2 (EZH2) inhibitor, with a Ki value <0.1 nM against mutant Y641N EZH2. Exhibits robust tumor growth inhibition.
Grouped product items
Product Name Price Stock Qty
PF-06821497 1mg
$320.00
In stock
PF-06821497 5mg
$960.00
In stock
PF-06821497 10mg
$1,600.00
In stock
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Biological Activity
Discription PF-06821497 (compound 23a) is a potent, selective and orally active Enhancer of Zeste Homolog 2 (EZH2) inhibitor, with a Ki value <0.1 nM against mutant Y641N EZH2. Exhibits robust tumor growth inhibition.
Product Information
Catalog Num A21388
Formula C22H24Cl2N2O5
Molecular Weight 467.34
CAS Number 1844849-10-0
SMILES COC1=C(CN2CCC(C(Cl)=CC([C@H](OC)C3COC3)=C4Cl)=C4C2=O)C(NC(C)=C1)=O
Synonyms PF06821497, PF 06821497
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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