TGR-1202 (Umbralisib)

Catalog No.: A16277
PI3Kδ inhibitor
TGR-1202 is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.
Grouped product items
Product Name Price Stock Qty
TGR-1202 5mg
$120.00
In stock
TGR-1202 10mg
$220.00
In stock
TGR-1202 50mg
$580.00
In stock
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Biological Activity
Discription TGR-1202 is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.
Targets
Target Value
Product Information
Catalog Num A16277
Formula C31H24F3N5O3
Molecular Weight 571.55
CAS Number 1532533-67-7
SMILES CC(C)OC1=C(C=C(C=C1)C2=NN(C3=C2C(=NC=N3)N)C(C)C4=C(C(=O)C5=C(O4)C=CC(=C5)F)C6=CC(=CC=C6)F)F
Synonyms RP5264, TGR1202, TGR 1202, RP-5264, RP 5264
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro (25°C) DMSO Warmed: 92 mg/mL (160.96 mM)
Water Insoluble
Ethanol Warmed: 6 mg/mL
In vivo 2% DMSO+30% PEG 300+2% Tween 80+H2O 2 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.5 mL 87.48 mL 174.96 mL
0.5 mM 3.5 mL 17.5 mL 34.99 mL
1 mM 1.75 mL 8.75 mL 17.5 mL
5 mM 0.35 mL 1.75 mL 3.5 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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