UPGL00004

Catalog No.: A19047
GAC inhibitor
UPGL00004 is a potent allosteric glutaminase C (GAC) inhibitor (IC50=29 nM; Kd=27 nM). UPGL00004 strongly inhibits the proliferation of highly aggressive triple-negative breast cancer cell lines.
Grouped product items
Product Name Price Stock Qty
UPGL00004 5mg
$350.00
In stock
UPGL00004 10mg
$650.00
In stock
UPGL00004 50mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500

Important Notice: For research use only. We do not sell to patients.

Not your Region? View all Distributors

Adooq Products cited in reputable paper
Biological Activity
Discription UPGL00004 is a potent allosteric glutaminase C (GAC) inhibitor (IC50=29 nM; Kd=27 nM). UPGL00004 strongly inhibits the proliferation of highly aggressive triple-negative breast cancer cell lines.
Product Information
Catalog Num A19047
Formula C25H26N8O2S2
Molecular Weight 534.66
CAS Number 1890169-95-5
SMILES O=C(NC1=NN=C(N2CCC(NC3=NN=C(NC(CC4=CC=CC=C4)=O)S3)CC2)S1)CC5=CC=CC=C5
Synonyms UPGL 00004, UPGL-00004
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 22 mg/mL (41.14 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.7 mL 93.52 mL 187.03 mL
0.5 mM 3.74 mL 18.7 mL 37.41 mL
1 mM 1.87 mL 9.35 mL 18.7 mL
5 mM 0.37 mL 1.87 mL 3.74 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2

  • Calculator Reset
Keywords: buy UPGL00004 | UPGL00004 Supplier | purchase UPGL00004 | UPGL00004 cost | UPGL00004 manufacturer | order UPGL00004 | UPGL00004 distributor | buy 1890169-95-5 | 1890169-95-5 Supplier | purchase 1890169-95-5 | 1890169-95-5 cost | 1890169-95-5 manufacturer | order 1890169-95-5 | 1890169-95-5 distributor