ERK5-IN-2
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | ERK5-IN-2 is an orally active, sub-micromolar, selective ERK5 inhibitor with IC50s of 0.82 μM, 3 μM for ERK5 and ERK5 MEF2D, respectively. | ||
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Targets |
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Catalog Num | A18871 |
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Formula | C17H11BrFN3O2 |
Molecular Weight | 388.19 |
CAS Number | 1888305-96-1 |
SMILES | FC1=CC=CC(Br)=C1C(C2=CNC(C(NC3=CC=CN=C3)=O)=C2)=O |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 66 mg/mL (170.02 mM) | |
Water | Insoluble | ||
Ethanol | 3 mg/mL (7.72 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 25.76 mL | 128.8 mL | 257.61 mL |
0.5 mM | 5.15 mL | 25.76 mL | 51.52 mL |
1 mM | 2.58 mL | 12.88 mL | 25.76 mL |
5 mM | 0.52 mL | 2.58 mL | 5.15 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2