GSK-2193874

Catalog No.: A14201
TRPV4 blocker
GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.
Grouped product items
Product Name Price Stock Qty
GSK-2193874 10mg
$130.00
In stock
GSK-2193874 25mg
$260.00
In stock
GSK-2193874 50mg
$425.00
In stock
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Biological Activity
Discription GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.
Product Information
Catalog Num A14201
Formula C37H38BrF3N4O
Molecular Weight 691.62
CAS Number 1336960-13-4
SMILES C1CCN(CC1)C2CCN(CC2)CC3=C(N=C4C=C(C=CC4=C3C(=O)NC5(CC5)C6=CC=CC=C6)Br)C7=CC(=CC=C7)C(F)(F)F
Synonyms GSK 2193874, GSK2193874
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 95 mg/mL (137.35 mM)
Water Insoluble
Ethanol Warmed: 48 mg/mL (69.4 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.46 mL 72.29 mL 144.59 mL
0.5 mM 2.89 mL 14.46 mL 28.92 mL
1 mM 1.45 mL 7.23 mL 14.46 mL
5 mM 0.29 mL 1.45 mL 2.89 mL
Useful Calculator

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