EPZ011989

Catalog No.: A15544
EZH2 Inhibitor
EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.
Grouped product items
Product Name Price Stock Qty
EPZ011989 5mg
$55.00
In stock
EPZ011989 10mg
$85.00
In stock
EPZ011989 25mg
$140.00
In stock
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Biological Activity
Discription EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.
Product Information
Catalog Num A15544
Formula C35H51N5O4
Molecular Weight 605.81
CAS Number 1598383-40-4
SMILES CCN(C1CCC(CC1)N(C)CCOC)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C#CCN4CCOCC4
Synonyms EPZ-011989, EPZ 011989
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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