DNA-PK

Catalog No.Inhibitor Name DNA-PKOther
A10726PI-103
**
p110α,p110δ,p110β
A11098NU7441
***
mTOR,PI3K
A10729PIK-75
****
p110α,p110γ,p110δ
A12752NU7026
*
PI3K
A11207PP121
**
PDGFR,Hck,VEGFR
A13224KU-0060648
***
PI3Kδ,PI3Kβ,PI3Kα
A11778Compound 401
*
mTOR,PI3K
A13328ETP-46464
***
ATM, ATR, PI3Kα, mTOR
A15779CC-115
***
mTOR

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. PIK-75

    Catalog No. A10729
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    PI3K Inhibitor
    PIK-75 is an imidazopyridine that selectively inhibits p110α with an IC50 value of 5.8 nM.2 It inhibits p110γ and p110β considerably less effectively with IC50 values of 0.076 µM and 1.3 µM, respectively. Learn More

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