EHT 1864

Catalog No.: A13886

Rac family GTPase inhibitor

EHT 1864

EHT 1864 Chemical Structure

CAS NO. 754240-09-0

EHT 1864 is an antiproliferative chemical shown to inhibit Rac family GTPases.

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10 mg
25 mg
50 mg
10mM * 1mL in DMSO
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Kakoki M, .et al. Engulfment and cell motility protein 1 potentiates diabetic cardiomyopathy via Rac-dependent and Rac-independent ROS production, JCI Insight, 2019, Jun 20;4(12) PMID: 31217360

Biological Activity

EHT 1864 is an antiproliferative chemical shown to inhibit Rac family GTPases.
Rac1 Rac1b Rac2 Rac3
40 nM(Kd)50 nM(Kd)60 nM(Kd)250 nM(Kd)
In vitro DMSO Warmed: 90 mg/mL (154.77 mM)
Water 90 mg/mL (154.77 mM)
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.2 mL 85.99 mL 171.98 mL
0.5 mM 3.44 mL 17.2 mL 34.4 mL
1 mM 1.72 mL 8.6 mL 17.2 mL
5 mM 0.34 mL 1.72 mL 3.44 mL

*The above data is based on the productmolecular weight 581.47. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13886
Actions Inhibitor
CAS No. 754240-09-0
Formula C25H27F3N2O4S.2HCl
M. Wt 581.47
Solubility DMSO
Purity >98%
Synonyms EHT-1864, EHT1864

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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