GSK-3787

Catalog No.: A12391

PPAR antagonist

GSK-3787 Chemical Structure

CAS NO. 188591-46-0

GSK-3787 is a potent and selective peroxisome proliferator-activated receptor δ (PPARδ) antagonist (pIC50 = 6.6).

Availability: In stock

Package Price Qty
10 mg
$70.00
25 mg
$140.00
50 mg
$220.00
100 mg
$380.00
10mM * 1mL in DMSO
$86.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GSK-3787 is a potent and selective peroxisome proliferator-activated receptor δ (PPARδ) antagonist (pIC50 = 6.6).
In vitro DMSO 79 mg/mL (201.13 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.46 mL 127.3 mL 254.6 mL
0.5 mM 5.09 mL 25.46 mL 50.92 mL
1 mM 2.55 mL 12.73 mL 25.46 mL
5 mM 0.51 mL 2.55 mL 5.09 mL

*The above data is based on the productmolecular weight 392.78. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12391
Actions Antagonist
M. Wt 392.78
Formula C15H12ClF3N2O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 188591-46-0
Synonyms GSK3787, GSK 3787
SMILES C1=CC(=CC=C1C(=O)NCCS(=O)(=O)C2=NC=C(C=C2)C(F)(F)F)Cl

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