GSK 525762A (I-BET-762)

Catalog No.: A11440

BET inhibitor

GSK 525762A (I-BET-762)

GSK 525762A (I-BET-762) Chemical Structure

CAS NO. 1260907-17-2

GSK-525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family

Availability: In stock

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5 mg
10 mg
25 mg
50 mg
10mM * 1mL in DMSO
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Biological Activity

GSK-525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family
BET proteins (Cell-free assay)
35 nM
In vitro DMSO 84 mg/mL (198.15 mM)
Water <1 mg/mL (<1 mM)
Ethanol 84 mg/mL (198.15 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.59 mL 117.95 mL 235.9 mL
0.5 mM 4.72 mL 23.59 mL 47.18 mL
1 mM 2.36 mL 11.8 mL 23.59 mL
5 mM 0.47 mL 2.36 mL 4.72 mL

*The above data is based on the productmolecular weight 423.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11440
Actions Inhibitor
M. Wt 423.9
Formula C22H22ClN5O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1260907-17-2
Synonyms GSK-525762A, GSK525762A
SMILES CCNC(=O)C[[email protected]]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C

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