Total item
Cart Subtotal
$0.00 Customer Appreciation Sale.
15% off with promo code "APPRECIATION2023" on check out or purchase order
Biological Activity
GSK-525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family
Targets
| BET proteins (Cell-free assay) | ||||
| 35 nM |
| In vitro | DMSO | 72 mg/mL (169.84 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 36 mg/mL (84.92 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.59 mL | 117.95 mL | 235.9 mL |
| 0.5 mM | 4.72 mL | 23.59 mL | 47.18 mL |
| 1 mM | 2.36 mL | 11.8 mL | 23.59 mL |
| 5 mM | 0.47 mL | 2.36 mL | 4.72 mL |
*The above data is based on the productmolecular weight 423.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A11440 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1260907-17-2 |
| Formula | C22H22ClN5O2 |
| M. Wt | 423.9 |
| Purity | >98% |
| Synonyms | GSK-525762A, GSK525762A |
| SMILES | CCNC(=O)C[[email protected]]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
Datasheet
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy GSK 525762A (I-BET-762) | GSK 525762A (I-BET-762) Supplier | purchase | cost | manufacturer | order | distributor | buy 1260907-17-2| 1260907-17-2 Supplier | purchase 1260907-17-2 | 1260907-17-2 cost | 1260907-17-2 manufacturer | order 1260907-17-2 | 1260907-17-2 distributor
Contact information
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: [email protected]
Not your Region? View all Distributors
Adooq Quality Guarantee
We promise all products perform as described.