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GSK 525762A (I-BET-762)

Catalog No.: A11440

BET inhibitor

GSK 525762A (I-BET-762)

GSK 525762A (I-BET-762) Chemical Structure

CAS NO. 1260907-17-2

GSK-525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family

Availability: In stock

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5 mg
10 mg
25 mg
50 mg
10mM * 1mL in DMSO
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Biological Activity

GSK-525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family
BET proteins (Cell-free assay)
35 nM
In vitro DMSO 72 mg/mL (169.84 mM)
Water Insoluble
Ethanol Warmed: 36 mg/mL (84.92 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.59 mL 117.95 mL 235.9 mL
0.5 mM 4.72 mL 23.59 mL 47.18 mL
1 mM 2.36 mL 11.8 mL 23.59 mL
5 mM 0.47 mL 2.36 mL 4.72 mL

*The above data is based on the productmolecular weight 423.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11440
Actions Inhibitor
CAS No. 1260907-17-2
Formula C22H22ClN5O2
M. Wt 423.9
Purity >98%
Synonyms GSK-525762A, GSK525762A
SMILES CCNC(=O)C[[email protected]]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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