KX2-391

Catalog No.: A11177

Src inhibitor

KX2-391

KX2-391 Chemical Structure

CAS NO. 897016-82-9

KX2-391 is a novel non-ATP competitive substrate-pocket directed SRC inhibitor.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $70.00

Special Price $63.00

10 mg

Regular Price: $120.00

Special Price $108.00

50 mg

Regular Price: $470.00

Special Price $423.00

100 mg

Regular Price: $800.00

Special Price $720.00

10mM * 1mL in DMSO

Regular Price: $119.00

Special Price $107.10

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

KX2-391 is a novel non-ATP competitive substrate-pocket directed SRC inhibitor.

Targets
Src (HuH7) (Cell-free assay) Src (PLC/PRF/5) (Cell-free assay) Src (Hep 3B) (Cell-free assay) Src (Hep G2) (Cell-free assay)
9 nM(GI50)13 nM(GI50)26 nM(GI50)60 nM(GI50)
In vitro (25°C) DMSO 86 mg/mL (199.29 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.17 mL 115.87 mL 231.73 mL
0.5 mM 4.63 mL 23.17 mL 46.35 mL
1 mM 2.32 mL 11.59 mL 23.17 mL
5 mM 0.46 mL 2.32 mL 4.63 mL

*The above data is based on the productmolecular weight 431.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11177
Actions Inhibitor
M. Wt 431.53
Formula C26H29N3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 897016-82-9
Synonyms KX2391
SMILES C1COCCN1CCOC2=CC=C(C=C2)C3=CN=C(C=C3)CC(=O)NCC4=CC=CC=C4

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