Total item
Cart Subtotal
$0.00 nAChR
24 Item(s)
per page
-
PNU 282987
Catalog No. A11233 α7 nAChR agonistPNU 282987 (PNU-282,987)is a drug that acts as a potent and selective agonist for the α7 subtype of neural nicotinic acetylcholine receptors. Learn More -
(-)-(S)-B-973B
Catalog No. A18761 α7 nAChR modulator-)-(S)-B-973B is a potent allosteric agonist and positive allosteric modulator of α7 nAChR, with antinociceptive activity. Learn More -
Mecamylamine Hydrochloride
Catalog No. A17884 nAChR antagonistMecamylamine hydrochloride is a nAChR antagonist previously used to treat hypertension. It displays a wide variety of activities, including reducing depression-like behaviors in subjects with Tourette's syndrome and improving rates of smoking cessation. Learn More -
Benzethonium Chloride
Catalog No. A13653 nAChR inhibitorBenzethonium chloride is a potent inhibitor of nAChRs, it inhibits α4β2 nAChRs and α7 nAChRs with IC50 of 49 nM and 122 nM, respectively. Learn More -
GTS-21 (DMBX-A)
Catalog No. A15950 nAChR agonistGTS-21 dihydrochloride is a selective α7 nicotinic acetylcholine receptor agonist, has recently been established as a promising treatment for inflammation. Learn More -
EVP-6124 hydrochloride
Catalog No. A15087 nAChR InhibitorEVP-6124 hydrochloride is a novel partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs). EVP-6124 showed selectivity for α7 nAChRs and did not activate or inhibit heteromeric α4β2 nAChRs. Learn More -
EVP-6124 (Encenicline)
Catalog No. A15086 nAChR InhibitorEVP-6124 is a novel partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs); shows selectivity for α7 nAChRs and did not activate or inhibit heteromeric α4β2 nAChRs. Learn More -
A-582941
Catalog No. A13539 α7 nAChR agonistA-582941 is a selective AChR a7 partial agonist. It exhibits high affinity for both rat and human a7 receptors (Ki values are 10.8 and 16.7 nM, respectively). Learn More -
5-Iodo-A-85380 2HCl
Catalog No. A13639 nAChR agonist5-Iodo-A-85380 2HCl is a highly potent and subtype-selective agonist for the a4b2 and a6b2 nicotinic acetylcholine receptors. Learn More -
ABT-418 HCl
Catalog No. A13688 nAChR agonistABT-418 HCl is a neuronal nicotinic acetylcholine receptor agonist. Learn More -
Sofinicline (ABT-894, A-422894)
Catalog No. A13842 nAChR agonistSofinicline is a novel nicotinic acetylcholine receptor agonist in the treatment of attention-deficit/hyperactivity disorder. Learn More -
Ispronicline (TC-1734, AZD-3480)
Catalog No. A14183 nAChR agonistIspronicline is a neuronal nicotinic acetylcholine receptor partial agonist. Ispronicline is subtype-selective, binding primarily to the a4b2 subtype. It has antidepressant, nootropic and neuroprotective effects. Learn More -
A-867744
Catalog No. A11290 modulator of α7 nAChRsA-867744 is a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor. Learn More -
Tropisetron HCL
Catalog No. A14375 5-HT3 receptor antagonistTropisetron is a selective 5-HT3 receptor antagonist and α7-nicotinic receptor agonist with an IC50 of 70.1 ± 0.9 nM for 5-HT3 receptor. Learn More -
Methyllycaconitine citrate
Catalog No. A12681 Methyllycaconitine citrate is a potent antagonist for α7-containing neuronal nicotinic receptors (Ki = 1.4 nM). Interacts with α4β2 and α6β2 receptors at concentrations > 40 nM. Learn More -
Adiphenine HCl
Catalog No. A11716 AChR inhibitorAdiphenine HCl is a nicotinic receptor inhibitor with IC50 of 15 μM, used as an antispasmodic drug Learn More -
Varenicline
Catalog No. A10966 -
PNU-120596
Catalog No. A11203 Nicotinic (α7) Receptor ModulatorPNU-120596 is a positive allosteric modulator of α7 neuronal nicotinic acetylcholine receptors. Learn More -
BNC375
Catalog No. A18503 α7 nAChR ModulatorBNC375 is a Potent, Selective, and Orally Available Type I Positive Allosteric Modulator of α7 nAChRs. Learn More -
Bephenium hydroxynaphthoate
Catalog No. A17391 B-type AChR activatorBephenium hydroxynaphthoate is an anthelmintic agent formerly used in the treatment of hookworm infections and ascariasis; B-type AChR activator. Learn More -
CCMI
Catalog No. A21534 α7 nAChR-positive allosteric modulatorCCMI is a potent and selective α7 nAChR-positive allosteric modulator, does not bind to or activate α7 nAChRs via the orthosteric site, and causes significant positive modulation of agonist-induced currents at α7 nAChRs. Learn More -
Varenicline Hydrochloride
Catalog No. A21539 α4β2 nAChR partial agonistVarenicline Hydrochloride (CP 526555 hydrochloride) is a high affinity, selective α4β2 nicotine acetylcholine receptor (nAChR) partial agonist and full α7 nAChR agonist. Learn More -
Tebanicline hydrochloride
Catalog No. A21918 nAChR modulatorTebanicline hydrochloride (ABT594 hydrochloride) is a nAChR modulator with potent, orally effective analgesic activity. Learn More -
Bephenium
Catalog No. A21680 AChR activatorBephenium is an anthelmintic agent formerly used in the treatment of hookworm infections and ascariasis; B-type AChR activator. Learn More
24 Item(s)
per page
FILTER BY:
Shopping Options
- Actions
-
- Inhibitor (4)
- Agonist (9)
- Antagonist (2)
- Activator (2)
- Modulator (6)
Contact information
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: [email protected]
Not your Region? View all Distributors
Adooq Quality Guarantee
We promise all products perform as described.