PCI-34051

Catalog No.: A11152

HDAC inhibitor

PCI-34051

PCI-34051 Chemical Structure

CAS NO. 950762-95-5

PCI-34051 is a specific and potent histone deacetylase 8 (HDAC8) inhibitor, with >200-fold selectivity over the other HDAC isoforms.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $100.00

Special Price $90.00

25 mg

Regular Price: $200.00

Special Price $180.00

50 mg

Regular Price: $350.00

Special Price $315.00

100 mg

Regular Price: $660.00

Special Price $594.00

10mM * 1mL in DMSO

Regular Price: $60.00

Special Price $54.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

PCI-34051 is a specific and potent histone deacetylase 8 (HDAC8) inhibitor, with >200-fold selectivity over the other HDAC isoforms.
Targets
Target Value
HDAC8IC50: 10nM
HDAC6IC50: 2.9μM
HDAC1IC50: 4μM
HDAC10IC50: 13μM
HDAC2IC50: >50μM
HDAC3IC50: >50μM
In vitro (25°C) DMSO 59 mg/mL (199.1 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 33.75 mL 168.75 mL 337.5 mL
0.5 mM 6.75 mL 33.75 mL 67.5 mL
1 mM 3.37 mL 16.87 mL 33.75 mL
5 mM 0.67 mL 3.37 mL 6.75 mL

*The above data is based on the productmolecular weight 296.3 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A11152
Actions Inhibitor
M. Wt 296.3
Formula C17H16N2O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 950762-95-5
Synonyms PCI34051
SMILES COC1=CC=C(C=C1)CN2C=CC3=C2C=C(C=C3)C(=O)NO

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