PD153035 (HCl salt)

Catalog No.: A10702

EGFR inhibitor

PD153035 (HCl salt) Chemical Structure

CAS NO. 183322-45-4

PD153035 is an extremely potent and specific inhibitor of the tyrosine kinase activity of EGFR.

Availability: In stock

Package Price Qty
10 mg
$50.00
50 mg
$220.00
100 mg
$380.00
200 mg
$630.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

PD153035 is an extremely potent and specific inhibitor of the tyrosine kinase activity of EGFR.
Targets
EGFR (Cell-free assay) EGFR (Cell-free assay)
5.2 pM(Ki)5.2 pM(Ki)
In vitro (25°C) DMSO 0.5 mg/mL (1.26 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% Propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.21 mL 126.04 mL 252.08 mL
0.5 mM 5.04 mL 25.21 mL 50.42 mL
1 mM 2.52 mL 12.6 mL 25.21 mL
5 mM 0.5 mL 2.52 mL 5.04 mL

*The above data is based on the productmolecular weight 396.7 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10702
Actions Inhibitor
M. Wt 396.7
Formula C16H14BrN3O2.HCl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 183322-45-4
Synonyms ZM 252868, AG 1517, Tyrphostin AG 1517, SU 5271, PD-153035
SMILES COC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC(=CC=C3)Br)OC.Cl

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