Pelitinib (EKB-569)

Name: Pelitinib (EKB-569)
SKU: A10706
Price: 35 USD
Rating: 5 (1 reviews)

Catalog No.: A10706

EGFR inhibitor

Adooq's Pelitinib (EKB-569) has been cited by 1 publications

Pelitinib (EKB-569) is a 3-cyanoquinoline pan-ErbB tyrosine kinase inhibitor with potential antineoplastic activity.

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Grouped product items
Size	Price	Stock
5mg	$35.00	In stock
10mg	$55.00	In stock
25mg	$100.00	In stock
50mg	$125.00	In stock
100mg	$190.00	In stock
500mg	$485.00	In stock
*10mM 1mL in DMSO**	$120.00	In stock
Bulk Size	Bulk Discount

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Important Notice: For research use only. We do not sell to patients.

Data Sheet

SDS

Adooq Products cited in reputable paper

Adooq's Pelitinib (EKB-569) has been cited by 1 publications

Shi P, .et al. , Transl Oncol, 2019, Mar 8;12(5):705-713 PMID: 30856555

Biological Activity

Discription

Pelitinib (EKB-569) is a 3-cyanoquinoline pan-ErbB tyrosine kinase inhibitor with potential antineoplastic activity.

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

Product Information

Catalog Num	A10706
Formula	C24H23ClFN5O2
Molecular Weight	467.9
CAS Number	257933-82-7
SMILES	CCOC1=C(C=C2C(=C1)N=CC(=C2NC3=CC(=C(C=C3)F)Cl)C#N)NC(=O)/C=C/CN(C)C
Synonyms	WAY-EKB 569
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro	DMSO	12 mg/mL (25.64 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.37 mL	106.86 mL	213.72 mL
0.5 mM	4.27 mL	21.37 mL	42.74 mL
1 mM	2.14 mL	10.69 mL	21.37 mL
5 mM	0.43 mL	2.14 mL	4.27 mL

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