Rimonabant (SR141716)
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Important Notice: For research use only. We do not sell to patients.
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Discription | Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane. | ||
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Catalog Num | A11547 |
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Formula | C22H21Cl3N4O |
Molecular Weight | 463.79 |
CAS Number | 168273-06-1 |
SMILES | CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)Cl |
Synonyms | SR141716 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 22 mg/mL (47.43 mM) | |
Water | Insoluble | ||
Ethanol | 2 mg/mL | ||
In vivo | 30% PEG400+0.5% Tween80+5% propylene glycol | 28 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 21.56 mL | 107.81 mL | 215.61 mL |
0.5 mM | 4.31 mL | 21.56 mL | 43.12 mL |
1 mM | 2.16 mL | 10.78 mL | 21.56 mL |
5 mM | 0.43 mL | 2.16 mL | 4.31 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2