Rimonabant (SR141716)

Catalog No.: A11547

Rimonabant (SR141716) Chemical Structure

CAS NO. 168273-06-1

Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.

Availability: In stock

Package Price Qty
10 mg
$50.00
25 mg
$110.00
50 mg
$200.00
100 mg
$350.00
10mM * 1mL in DMSO
$87.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
Targets
hCB1 hCB2 ACAT
13.6 nM1.64 μM1.5 μM-2.9 μM
In vitro (25°C) DMSO 25 mg/mL (53.9 mM)
Water <1 mg/mL (<1 mM)
Ethanol 2 mg/mL (4.31 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.56 mL 107.81 mL 215.61 mL
0.5 mM 4.31 mL 21.56 mL 43.12 mL
1 mM 2.16 mL 10.78 mL 21.56 mL
5 mM 0.43 mL 2.16 mL 4.31 mL

*The above data is based on the productmolecular weight 463.79. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11547
Actions N/A
M. Wt 463.79
Formula C22H21Cl3N4O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 168273-06-1
Synonyms SR141716
SMILES CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)Cl

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