Rimonabant (SR141716)

Catalog No.: A11547

Rimonabant (SR141716)

Rimonabant (SR141716) Chemical Structure

CAS NO. 168273-06-1

Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $50.00

Special Price $40.00

25 mg

Regular Price: $110.00

Special Price $88.00

50 mg

Regular Price: $200.00

Special Price $160.00

100 mg

Regular Price: $350.00

Special Price $280.00

10mM * 1mL in DMSO

Regular Price: $87.00

Special Price $69.60

Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
Targets
hCB1 hCB2 ACAT
13.6 nM1.64 μM1.5 μM-2.9 μM
In vitro (25°C) DMSO 22 mg/mL (47.43 mM)
Water Insoluble
Ethanol 2 mg/mL
In vivo 30% PEG400+0.5% Tween80+5% propylene glycol 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.56 mL 107.81 mL 215.61 mL
0.5 mM 4.31 mL 21.56 mL 43.12 mL
1 mM 2.16 mL 10.78 mL 21.56 mL
5 mM 0.43 mL 2.16 mL 4.31 mL

*The above data is based on the productmolecular weight 463.79. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11547
CAS No. 168273-06-1
Formula C22H21Cl3N4O
M. Wt 463.79
Purity >98%
Synonyms SR141716
SMILES CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Rimonabant (SR141716) | Rimonabant (SR141716) Supplier | purchase | cost | manufacturer | order | distributor | buy 168273-06-1| 168273-06-1 Supplier | purchase 168273-06-1 | 168273-06-1 cost | 168273-06-1 manufacturer | order 168273-06-1 | 168273-06-1 distributor
Rewards