ROCK inhibitor

Catalog No.: A15225

ROCK inhibitor

ROCK inhibitor

ROCK inhibitor Chemical Structure

CAS NO. 867017-68-3

ROCK inhibitor is a highly potent inhibitor of human ROCK-1 and ROCK-2 isoenzymes with IC50 values of 0.6 and 1.1 nM, respectively.

Availability: In stock

Package Price Qty
5 mg
$300.00
10 mg
$450.00
50 mg
$1,100.00
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Biological Activity

ROCK inhibitor is a highly potent inhibitor of human ROCK-1 and ROCK-2 isoenzymes with IC50 values of 0.6 and 1.1 nM, respectively.
In vitro DMSO 77 mg/mL (191.16 mM)
Water Insoluble
Ethanol 2 mg/mL (4.96 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.83 mL 124.13 mL 248.27 mL
0.5 mM 4.97 mL 24.83 mL 49.65 mL
1 mM 2.48 mL 12.41 mL 24.83 mL
5 mM 0.5 mL 2.48 mL 4.97 mL

*The above data is based on the productmolecular weight 402.79. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15225
Actions Inhibitor
CAS No. 867017-68-3
Formula C18H13ClF2N6O
M. Wt 402.79
Purity >98%
Synonyms Rho-kinase inhibitor, Rho Kinase Inhibitor, ROCK
SMILES CC1=CNC2=NC=CC(=C12)OC3=C(C=C(C=C3F)NC4=CC(=NC(=N4)N)Cl)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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