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Products tagged with 'CYP2C9'

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  1. Apigenin

    Catalog No. A10081
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    Protein kinase inhibitor

    Apigenin, found in many plants, is a natural product belonging to the flavone class that is the aglycone of several naturally-occurring glycosides. Apigenin acts as a monoamine transporter activator, one of the few chemicals demonstrated to possess this property. Apigenin is a ligand for central benzodiazepine receptors that competitively inhibited the binding of flunitrazepam with a Ki of 4μM, exerting anxiolytic and slight sedative effects.

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  2. Avasimibe (CI-1011)

    Catalog No. A10102
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    CYP17 inhibitor
    Avasimibe (CI-1011) is an orally bioavailable Acyl-CoA:Cholesterol O-Acyltransferase (ACAT) inhibitor. Learn More
  3. Baicalein

    Catalog No. A10120
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    Lipoxygenase Inhibitor

    Baicalein is a flavonoid originally isolated from the roots of Scutellaria baicalensis Georgi. Baicalein inhibits lipid peroxidation, as assessed by production of TBARS, with an IC50 value of 5 µM.

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  4. Benzbromarone

    Catalog No. A16201
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    CYP2C9 inhibitor
    Benzbromarone is a CYP2C9 inhibitor, it binds to CYP2C9 with Ki value of 19.3 nM. Learn More
  5. Ticagrelor (AZD6140)

    Catalog No. A11238
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    P2Y12 antagonist
    Ticagrelor (AZD6140) is the first reversibly binding oral P2Y(12) receptor antagonist that blocks ADP-induced platelet aggregation. Learn More

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