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Products tagged with 'GABAA receptor'

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  1. (+)-Bicuculline

    Catalog No. A12590
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    GABAA antagonist
    (+)-Bicuculline is a classical GABAA antagonist. Learn More
  2. Apalutamide (ARN-509)

    Catalog No. A11923
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    Androgen Receptor inhibitor
    ARN-509 is an androgen receptor antagonist with potential antineoplastic activity. ARN-509 binds to AR in target tissues thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot be translocated to the nucleus. This prevents binding to and transcription of AR-responsive genes. Learn More
  3. Baicalin

    Catalog No. A10121
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    HIV-1 production Inhibitor
    Baicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors. Learn More
  4. Dihydromyricetin (Ampeloptin)

    Catalog No. A10252
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    Dihydropyrimidinase Inhibitor
    Dihydromyricetin (Ampelopsin (flavanol); Ampeloptin) is a natural antioxidant with good prospects. Learn More
  5. Flumazenil

    Catalog No. A10397
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    Benzodiazepine antagonist
    Flumazenil, an imidazobenzodiazepine derivative, antagonizes the actions of benzodiazepines on the central nervous system. Flumazenil competitively inhibits the activity at the benzodiazepine recognition site on the GABA/benzodiazepine receptor complex. Flumazenil is a weak partial agonist in some animal models of activity, but has little or no agonist activity in humans. Learn More
  6. Zolpidem

    Catalog No. A15288
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    Benzodiazepine agonist
    Zolpidem is an inhibitory neurotransmitter, by binding to GABAA receptors at the same location as benzodiazepines. Learn More

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