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Products tagged with 'Histamine H1 receptor'

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  1. Bepotastine Besilate

    Catalog No. A11340
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    Histamine Receptor antagonist
    Bepotastine Beslilate (Bepreve) is a histamine H1 receptor anatagonist. Learn More
  2. Brompheniramine

    Catalog No. A11699
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    Brompheniramine is a first-generation antihistamine. Brompheniramine works by acting as an antagonist of histamine H1 receptors. It also functions as a moderately effective anticholinergic agent, and is likely an antimuscarinic agent similar to other common antihistamines such as diphenhydramine. Learn More
  3. CarbinoxaMine Maleate

    Catalog No. A16129
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    histamine-H1 receptor blocking agent
    Carbinoxamine maleate is a histamine-H1 receptor blocking agent with antihistamine and anticholinergic properties. Learn More
  4. Chlorpheniramine maleate

    Catalog No. A10205
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    Chlorpheniramine maleate is a first-generation alkylamine antihistamine used in the prevention of the symptoms of allergic conditions such as rhinitis and urticaria. Learn More
  5. Clemastine fumarate

    Catalog No. A10226
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    Histamine Receptor antagonis
    Clemastine is a selective histamine H1 antagonist. It binds to the histamine H1 receptor, thus blocking the action of endogenous histamine, which leads to temporary relief of the negative symptoms caused by histamine. Learn More
  6. Diphenhydramine hcl

    Catalog No. A10318
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    Diphenhydramine is a first-generation antihistamine possessing anticholinergic, antitussive, antiemetic and sedative properties which is mainly used to treat allergies. Learn More
  7. Ebastine

    Catalog No. A14946
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    H1-histamine receptor antagonist
    Ebastine is a H1 antihistamine with low potential for causing drowsiness. Learn More
  8. Fexofenadine HCl

    Catalog No. A11859
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    COX inhibitor/histamine H1 receptor agonist
    Fexofenadine HCl is an antihistamine that inhibits Cox-1, Cox-2, and is a histamine H1 receptor agonist Learn More
  9. Lidocaine (Alphacaine)

    Catalog No. A10530
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    Lidocaine (Alphacaine) is an anasthetic and class Ib antiarrhythmic agent. Blocks voltage-gated sodium channels in the inactivated state. Learn More
  10. Loratadine

    Catalog No. A10538
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    Loratadine is a non-sedative antihistamine that inhibits histamine-induced activities of IL-6 and IL-8 secretion in endothelial cells. Loratadine is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM. Learn More
  11. Meclizine 2HCl

    Catalog No. A11700
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    Meclizine is a human pregnane X receptor (hPXR) agonist. It possesses anticholinergic, central nervous system depressant, and local anesthetic effects. Its antiemetic and antivertigo effects are not fully understood, but its central anticholinergic properties are partially responsible. Learn More
  12. Mizolastine

    Catalog No. A11724
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    Mizolastine is a second generation antihistamine agent with high affinity and specificity for histamine H1 receptors. Learn More
  13. Rupatadine Fumarate

    Catalog No. A12356
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    PAFR inhibitor/H1 receptor inhibitor
    Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively. Learn More

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