TRV130 (Oliceridine)

Catalog No.: A14337

μ-opioid receptor agonist

TRV130 (Oliceridine) Chemical Structure

CAS NO. 1401028-24-7

TRV130 is an opioid drug that is under evaluation in human clinical trials for the treatment of acute severe pain. TRV130 elicits robust G protein signaling, with potency and efficacy similar to morphine, but with far less ??-arrestin 2 recruitment and receptor internalization, it displays less adverse effects than morphine.

Availability: In stock

Package Price Qty
5 mg
$90.00
10 mg
$150.00
25 mg
$300.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

TRV130 is an opioid drug that is under evaluation in human clinical trials for the treatment of acute severe pain. TRV130 elicits robust G protein signaling, with potency and efficacy similar to morphine, but with far less ??-arrestin 2 recruitment and receptor internalization, it displays less adverse effects than morphine.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.64 mL 118.2 mL 236.4 mL
0.5 mM 4.73 mL 23.64 mL 47.28 mL
1 mM 2.36 mL 11.82 mL 23.64 mL
5 mM 0.47 mL 2.36 mL 4.73 mL

*The above data is based on the productmolecular weight 423.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14337
Actions Agonist
M. Wt 423.01
Formula C22H31ClN2O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1401028-24-7
Synonyms TRV 130, TRV-130
SMILES COC1=C(SC=C1)CNCC[[email protected]]2(CCOC3(C2)CCCC3)C4=CC=CC=N4

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