Product Data Sheet

AR-C155858

Catalog No. A11293

main product photo
AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.
Adooq's AR-C155858 has been cited by 6 publications
  • Charlotte Petersen, .et al. , Sci Rep, 2017, 7: 13101 PMID: 29026134
  • Kong SC, .et al. , Pancreas, 2016, Aug;45(7):1036-47 PMID: 26765963
  • Anne Poder, .et al. , Mol Cancer, 2016, 15: 45 PMID: 27266704
  • Eumorphia G. Konstantakou, .et al. , Mol Cancer, 2015, 14: 135 PMID: 26198749
  • Álvarez Z, .et al. , Biomaterials., 2014, 35(17):4769-81 PMID: 24636215
  • Álvarez Z, .et al. , Cereb Cortex., 2014, 26(3):1046-58 PMID: 25452568
    • Chemical Information
    Catalog Num A11293
    M. Wt 461.5
    Formula C21H27N5O5S
    Purity >98%
    Storage at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base)
    CAS No. 496791-37-8
    Synonyms AR-C 155858
    SMILES CC1=C(C(=NN1)C)CC2=C(C3=C(S2)N(C(=O)N(C3=O)C)CC(C)C)C(=O)N4C[C@@H](CO4)O
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
    Biological Activity
    Discription AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.
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    SHIPPING AND STORAGE
    Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.