Product Data Sheet

ENOblock (AP-III-a4)

Catalog No. A11840

main product photo
ENOblock (AP-III-a4) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo.
Adooq's ENOblock (AP-III-a4) has been cited by 2 publications
  • Rachel Polcyn, .et al. , Neurochem Int, 2020, Jul 7;104788 PMID: 32650031
  • Yakarsonmez S, .et al. , Mol Divers, 2019, Nov 21 PMID: 31754915
  • Chemical Information
    Catalog NumA11840
    M. Wt594.72
    FormulaC31H43FN8O3
    Purity>98%
    Storageat -20 °C 3 years (powder form); at -20 °C 6 months (Solution base)
    CAS No.1177827-73-4
    Synonyms
    SMILESC1CCC(CC1)CNC2=NC(=NC(=N2)NCC3=CC=C(C=C3)F)NC4=CC=C(C=C4)CC(=O)NCCOCCOCCN
    Biological Activity
    DescriptionENOblock (AP-III-a4) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo.
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    SHIPPING AND STORAGE
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