Product Data Sheet

Elacridar (GF120918)

Catalog No. A12324

main product photo
Elacridaris a prototypical BCRP inhibitor which inhibits the Bcrp1-mediated transport.
Adooq's Elacridar (GF120918) has been cited by 1 publications
  • Leo Shen, .et al. , Sci Rep, 2021, Sep 16;11(1):18516 PMID: 34531456
  • Chemical Information
    Catalog NumA12324
    M. Wt563.64
    FormulaC34H33N3O5
    Purity>98%
    Storageat -20 °C 3 years (powder form); at -20 °C 6 months (Solution base)
    CAS No.143664-11-3
    Synonyms
    SMILESCOC1=CC=CC2=C1NC3=C(C2=O)C=CC=C3C(=O)NC4=CC=C(C=C4)CCN5CCC6=CC(=C(C=C6C5)OC)OC
    Biological Activity
    DescriptionElacridaris a prototypical BCRP inhibitor which inhibits the Bcrp1-mediated transport.
    Targets
    TargetValue
    Solubility
    In vitro (25°C) DMSOWarmed: 7 mg/mL (12.42 mM)
    WaterInsoluble
    EthanolInsoluble
    In vivo 4% DMSO+30% PEG 300+5% Tween 80+ddH2O 1 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass1 mg5 mg10 mg
    0.1 mM17.74 mL88.71 mL177.42 mL
    0.5 mM3.55 mL17.74 mL35.48 mL
    1 mM1.77 mL8.87 mL17.74 mL
    5 mM0.35 mL1.77 mL3.55 mL
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    SHIPPING AND STORAGE
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