Product Data Sheet
Thermopsidine
Catalog No. A13859
Thermopsidine is a selective partial agonist of the α4β2 and α6β2 nicotinic acetylcholine receptors (nAChRs), exhibiting an EC50 value of 2.2 μM for the α4β2 subtype. This compound is valuable for studying cholinergic signaling pathways and exploring potential therapeutic avenues in neurodegenerative diseases and addiction research. Its specific targeting of nAChRs makes it a useful tool for evaluating receptor function and pharmacology.
Chemical Information
| Catalog Num | A13859 |
|---|---|
| M. Wt | 406.52 |
| Formula | C24H30N4O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 492-02-4 |
| Synonyms | CC4 |
| SMILES | [H][C@@]12CN3C([C@@](C2)([H])CN(C1)CCN4C[C@](C5)([H])C(N6C[C@]5([H])C4)=CC=CC6=O)=CC=CC3=O |
Biological Activity
| Description | Thermopsidine is a selective partial agonist of the α4β2 and α6β2 nicotinic acetylcholine receptors (nAChRs), exhibiting an EC50 value of 2.2 μM for the α4β2 subtype. This compound is valuable for studying cholinergic signaling pathways and exploring potential therapeutic avenues in neurodegenerative diseases and addiction research. Its specific targeting of nAChRs makes it a useful tool for evaluating receptor function and pharmacology. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
