Product Data Sheet

Amezinium methylsulfate

Catalog No. A18103

main product photo
Amezinium Metilsulfate, also known as Regulton and LU-1631, is a norepinephrine reuptake inhibitor which exclusively affects postganglionic sympathetic neurons. Amezinium Metilsulfate is used to treat hypotension.
Chemical Information
Catalog Num A18103
M. Wt 313.33
Formula C12H15N3O5S
Purity >98%
Storage at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base)
CAS No. 30578-37-1
Synonyms Amezinium Metilsulfate; LU-1631; LU 1631; LU1631; Regulton; Risumic
SMILES COC1=CC(N)=CN=[N+]1C2=CC=CC=C2.O=S(OC)([O-])=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Biological Activity
Discription Amezinium Metilsulfate, also known as Regulton and LU-1631, is a norepinephrine reuptake inhibitor which exclusively affects postganglionic sympathetic neurons. Amezinium Metilsulfate is used to treat hypotension.
Solubility
In vitro DMSO 60 mg/mL (191.49 mM)
Water 31 mg/mL (98.93 mM)
Ethanol 5 mg/mL (15.95 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 31.92 mL 159.58 mL 319.15 mL
0.5 mM 6.38 mL 31.92 mL 63.83 mL
1 mM 3.19 mL 15.96 mL 31.92 mL
5 mM 0.64 mL 3.19 mL 6.38 mL
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SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.