Product Data Sheet
Linagliptin-d3-1
Catalog No. A26872
Linagliptin-d3-1 is a deuterium-labeled analog of Linagliptin, a highly potent and selective inhibitor of dipeptidyl peptidase-4 (DPP-4) with an IC50 of 1 nM. This isotope-labeled compound is primarily utilized in pharmacokinetic studies and metabolic research to trace the pharmacological pathways of DPP-4 inhibitors in various biological systems. Its unique isotopic signature allows for enhanced detection and quantification in analytical applications, facilitating insights into drug metabolism and efficacy.
Chemical Information
| Catalog Num | A26872 |
|---|---|
| M. Wt | 475.56 |
| Formula | C25H25D3N8O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1398044-48-8 |
| Synonyms | BI 1356-d3-1 |
| SMILES | O=C1N(C2=C(C(N1CC3=NC(C)=C4C=CC=CC4=N3)=O)N(CC#CC([2H])([2H])[2H])C(N5CCC[C@@H](N)C5)=N2)C |
Biological Activity
| Description | Linagliptin-d3-1 is a deuterium-labeled analog of Linagliptin, a highly potent and selective inhibitor of dipeptidyl peptidase-4 (DPP-4) with an IC50 of 1 nM. This isotope-labeled compound is primarily utilized in pharmacokinetic studies and metabolic research to trace the pharmacological pathways of DPP-4 inhibitors in various biological systems. Its unique isotopic signature allows for enhanced detection and quantification in analytical applications, facilitating insights into drug metabolism and efficacy. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
