Product Data Sheet
DS-9300
Catalog No. A29185
DS-9300 is a selective inhibitor of the EP300/CBP histone acetyltransferases (HATs) with a potent IC50 value of 28 nM. This compound demonstrates significant anticancer activity and is applicable in prostate cancer research, providing valuable insights into the mechanisms of acetylation in tumorigenesis. DS-9300 serves as a critical tool for studying the role of HATs in cancer progression and therapeutic resistance.
Chemical Information
| Catalog Num | A29185 |
|---|---|
| M. Wt | 501.50 |
| Formula | C25H26F3N5O3 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2259641-46-6 |
| Synonyms | |
| SMILES | COC1=CC=C(C=C1)C2(CCC(F)(CC2)F)C(N3C[C@@H](C[C@@H]3C(NC4=NC5=C(NN=C5)C=C4)=O)F)=O |
Biological Activity
| Description | DS-9300 is a selective inhibitor of the EP300/CBP histone acetyltransferases (HATs) with a potent IC50 value of 28 nM. This compound demonstrates significant anticancer activity and is applicable in prostate cancer research, providing valuable insights into the mechanisms of acetylation in tumorigenesis. DS-9300 serves as a critical tool for studying the role of HATs in cancer progression and therapeutic resistance. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
