Product Data Sheet
5-HT7R antagonist 4
Catalog No. A29371
5-HT7R antagonist 4 is a selective antagonist of the 5-HT7 receptor, exhibiting a binding affinity of Ki = 2.6 nM, while demonstrating lower affinity for the 5-HT1A receptor (Ki = 476 nM). This compound serves as a valuable tool for investigating the role of 5-HT7 receptors in neurological disorders and may contribute to the development of therapeutic strategies targeting these pathways. Its pharmacological profile makes it suitable for research applications focused on serotonin-related signaling and neurodegenerative diseases.
Chemical Information
| Catalog Num | A29371 |
|---|---|
| M. Wt | 268.35 |
| Formula | C17H20N2O |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1386927-90-7 |
| Synonyms | |
| SMILES | COC1=CC=C(C=C1)C2=CC=CC=C2N3CCNCC3 |
Biological Activity
| Description | 5-HT7R antagonist 4 is a selective antagonist of the 5-HT7 receptor, exhibiting a binding affinity of Ki = 2.6 nM, while demonstrating lower affinity for the 5-HT1A receptor (Ki = 476 nM). This compound serves as a valuable tool for investigating the role of 5-HT7 receptors in neurological disorders and may contribute to the development of therapeutic strategies targeting these pathways. Its pharmacological profile makes it suitable for research applications focused on serotonin-related signaling and neurodegenerative diseases. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
