Carpindolol
Catalog No. A29501

Carpindolol is a selective antagonist of the 5-HT1B receptor and an agonist of the 5-HT1D receptor, demonstrating a pKd of 8.53 and pKB of 8.0 for its antagonistic activity, as well as a pEC50 of 5.91 for its agonistic effects. This compound has significant implications in neuropharmacology research, particularly in studies investigating serotonin receptor dynamics and related pathways. It serves as a valuable tool for exploring the modulation of neurotransmitter systems and their physiological roles.
Chemical Information
| Catalog Num | A29501 |
|---|---|
| M. Wt | 348.44 |
| Formula | C19H28N2O4 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 39731-05-0 |
| Synonyms | SDZ21009 |
| SMILES | O=C(C(N1)=CC2=C1C=CC=C2OCC(O)CNC(C)(C)C)OC(C)C |
Biological Activity
| Description | Carpindolol is a selective antagonist of the 5-HT1B receptor and an agonist of the 5-HT1D receptor, demonstrating a pKd of 8.53 and pKB of 8.0 for its antagonistic activity, as well as a pEC50 of 5.91 for its agonistic effects. This compound has significant implications in neuropharmacology research, particularly in studies investigating serotonin receptor dynamics and related pathways. It serves as a valuable tool for exploring the modulation of neurotransmitter systems and their physiological roles. |
|---|
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Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.


