Product Data Sheet
5-HT2CR agonist 1
Catalog No. A29603
5-HT2CR agonist 1 is a selective partial agonist of the 5-HT2C receptor, displaying an effective maximum response (Emax) of 71.09% and an EC50 of 121.5 nM. This compound has been shown to exhibit specificity, with no activity towards 5-HT2A or 5-HT2B receptors. Furthermore, it demonstrates no recruitment activity for β-arrestin and minimal inhibition of hERG channels at 10 μM. This profile makes 5-HT2CR agonist 1 a valuable tool for research in neuropharmacology and receptor signaling pathways.
Chemical Information
| Catalog Num | A29603 |
|---|---|
| M. Wt | 235.71 |
| Formula | C13H14ClNO |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1216074-15-5 |
| Synonyms | |
| SMILES | ClC1=CC=C2C=CC3(OC2=C1)CCNCC3 |
Biological Activity
| Description | 5-HT2CR agonist 1 is a selective partial agonist of the 5-HT2C receptor, displaying an effective maximum response (Emax) of 71.09% and an EC50 of 121.5 nM. This compound has been shown to exhibit specificity, with no activity towards 5-HT2A or 5-HT2B receptors. Furthermore, it demonstrates no recruitment activity for β-arrestin and minimal inhibition of hERG channels at 10 μM. This profile makes 5-HT2CR agonist 1 a valuable tool for research in neuropharmacology and receptor signaling pathways. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
