Product Data Sheet
CSP-2503
Catalog No. A29643
CSP-2503 is a highly selective agonist of the 5-HT1A receptor, exhibiting an EC50 of 0.15 μM and a Ki value of 4.1 nM. This compound demonstrates significant selectivity against α1-adrenoceptors, 5-HT4 receptors, and benzodiazepine receptors, with Ki values exceeding 1000 nM. CSP-2503 reduces cAMP levels in vitro and displays anxiolytic effects in vivo, making it a valuable tool for investigating anxiety-related disorders.
Chemical Information
| Catalog Num | A29643 |
|---|---|
| M. Wt | 378.48 |
| Formula | C22H26N4O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 581813-10-7 |
| Synonyms | |
| SMILES | C(N1CCN(C=2C3=C(C=CC2)C=CC=C3)CC1)N4C(=O)[C@]5(N(C(=O)C4)CCC5)[H] |
Biological Activity
| Description | CSP-2503 is a highly selective agonist of the 5-HT1A receptor, exhibiting an EC50 of 0.15 μM and a Ki value of 4.1 nM. This compound demonstrates significant selectivity against α1-adrenoceptors, 5-HT4 receptors, and benzodiazepine receptors, with Ki values exceeding 1000 nM. CSP-2503 reduces cAMP levels in vitro and displays anxiolytic effects in vivo, making it a valuable tool for investigating anxiety-related disorders. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
