Product Data Sheet
5-HT2A/5-HT2C inverse agonist 1
Catalog No. A29685
5-HT2A/5-HT2C inverse agonist 1 functions as a potent dual inverse agonist at the 5-HT2A and 5-HT2C receptors, demonstrating minimal hERG channel inhibition to mitigate cardiovascular risks. This compound exhibits significant antipsychotic effects in the MK-801-induced mouse model, making it a valuable tool for the investigation of psychotic disorders. It is particularly relevant for studies aiming to elucidate the molecular mechanisms underlying psychosis and for the development of new therapeutic strategies.
Chemical Information
| Catalog Num | A29685 |
|---|---|
| M. Wt | 425.57 |
| Formula | C24H35N5O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2718990-76-0 |
| Synonyms | |
| SMILES | CN(C=C1)N=C1CN([C@@H]2C3(CN(CC2)C)CC3)C(NCC4=CC=C(C=C4)OCCC)=O |
Biological Activity
| Description | 5-HT2A/5-HT2C inverse agonist 1 functions as a potent dual inverse agonist at the 5-HT2A and 5-HT2C receptors, demonstrating minimal hERG channel inhibition to mitigate cardiovascular risks. This compound exhibits significant antipsychotic effects in the MK-801-induced mouse model, making it a valuable tool for the investigation of psychotic disorders. It is particularly relevant for studies aiming to elucidate the molecular mechanisms underlying psychosis and for the development of new therapeutic strategies. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
