Product Data Sheet
Mazapertine
Catalog No. A29721
Mazapertine is an orally active antipsychotic agent primarily targeting dopamine D2, D3, and D4 receptors with high affinity (Ki values < 3 nM). Additionally, it exhibits significant binding to serotonin 5-HT1A receptors (Ki = 1.7 nM) and α1-adrenergic receptors (Ki = 1.3 nM). This compound is valuable for research into neurological diseases, particularly in the context of antipsychotic drug development and neuropharmacology studies.
Chemical Information
| Catalog Num | A29721 |
|---|---|
| M. Wt | 421.58 |
| Formula | C26H35N3O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 134208-17-6 |
| Synonyms | |
| SMILES | CC(C)OC1=C(N2CCN(CC3=CC(C(N4CCCCC4)=O)=CC=C3)CC2)C=CC=C1 |
Biological Activity
| Description | Mazapertine is an orally active antipsychotic agent primarily targeting dopamine D2, D3, and D4 receptors with high affinity (Ki values < 3 nM). Additionally, it exhibits significant binding to serotonin 5-HT1A receptors (Ki = 1.7 nM) and α1-adrenergic receptors (Ki = 1.3 nM). This compound is valuable for research into neurological diseases, particularly in the context of antipsychotic drug development and neuropharmacology studies. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
