Product Data Sheet
PF-03246799 monohydrochloride
Catalog No. A29725
PF-03246799 monohydrochloride is a potent and selective agonist of the 5-HT2C receptor, exhibiting an EC50 of 190 nM and a Ki of 160 nM. This compound demonstrates a high selectivity for the 5-HT2C receptor compared to the 5-HT2A and 5-HT2B receptors. PF-03246799 monohydrochloride is primarily utilized in research focused on stress urinary incontinence (SUI) and may contribute to further understanding of serotonergic modulation in related conditions.
Chemical Information
| Catalog Num | A29725 |
|---|---|
| M. Wt | 275.78 |
| Formula | C15H18ClN3 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1613666-08-2 |
| Synonyms | |
| SMILES | C12=NC(CC3=CC=CC=C3)=NC=C1CCNCC2.Cl |
Biological Activity
| Description | PF-03246799 monohydrochloride is a potent and selective agonist of the 5-HT2C receptor, exhibiting an EC50 of 190 nM and a Ki of 160 nM. This compound demonstrates a high selectivity for the 5-HT2C receptor compared to the 5-HT2A and 5-HT2B receptors. PF-03246799 monohydrochloride is primarily utilized in research focused on stress urinary incontinence (SUI) and may contribute to further understanding of serotonergic modulation in related conditions. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
