Product Data Sheet
Pelanserin
Catalog No. A29842
Pelanserin is an orally active antihypertensive agent that primarily functions as a potent 5-HT2 receptor antagonist. It effectively inhibits α-adrenergic receptor activity, showcasing an ED50 value of 0.03 μg/mL. Additionally, Pelanserin demonstrates vasodilatory properties with an ED100 of 5 μg. This compound is valuable for research applications focused on hypertension, proving effective in hypertensive rodent models and renal hypertensive dog breeds.
Chemical Information
| Catalog Num | A29842 |
|---|---|
| M. Wt | 364.44 |
| Formula | C21H24N4O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2208-51-7 |
| Synonyms | |
| SMILES | O=C1NC2=C(C(N1CCCN3CCN(CC3)C4=CC=CC=C4)=O)C=CC=C2 |
Biological Activity
| Description | Pelanserin is an orally active antihypertensive agent that primarily functions as a potent 5-HT2 receptor antagonist. It effectively inhibits α-adrenergic receptor activity, showcasing an ED50 value of 0.03 μg/mL. Additionally, Pelanserin demonstrates vasodilatory properties with an ED100 of 5 μg. This compound is valuable for research applications focused on hypertension, proving effective in hypertensive rodent models and renal hypertensive dog breeds. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
