Anpirtoline
Catalog No. A29929

Anpirtoline is a potent agonist of the 5-HT1B receptor, exhibiting a Ki of 28 nM for this target, alongside 150 nM for 5-HT1A and 1.49 μM for 5-HT2 receptors. This compound demonstrates notable serotonergic activity and has been linked to antinociceptive and antidepressant-like effects. Anpirtoline is primarily utilized in research to explore its potential therapeutic applications in mood disorders and pain management.
Chemical Information
| Catalog Num | A29929 |
|---|---|
| M. Wt | 228.74 |
| Formula | C10H13ClN2S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 98330-05-3 |
| Synonyms | D-16949 |
| SMILES | ClC1=NC(SC2CCNCC2)=CC=C1 |
Biological Activity
| Description | Anpirtoline is a potent agonist of the 5-HT1B receptor, exhibiting a Ki of 28 nM for this target, alongside 150 nM for 5-HT1A and 1.49 μM for 5-HT2 receptors. This compound demonstrates notable serotonergic activity and has been linked to antinociceptive and antidepressant-like effects. Anpirtoline is primarily utilized in research to explore its potential therapeutic applications in mood disorders and pain management. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.


