Product Data Sheet
Cyamemazine-d6
Catalog No. A29983
Cyamemazine-d6 is a deuterated derivative of Cyamemazine, a neuroleptic agent characterized by its phenothiazine structure. This compound functions primarily as a potent antagonist of the 5-HT3 (Ki of 12 nM), 5-HT2A (Ki of 1.5 nM), and 5-HT2C (Ki of 75 nM) receptors, exhibiting notable anxiolytic and antipsychotic properties. Cyamemazine-d6 serves as a valuable stable isotope for studies involving pharmacokinetics, trace labeling, and metabolic research in the context of psychiatric disorders.
Chemical Information
| Catalog Num | A29983 |
|---|---|
| M. Wt | 329.49 |
| Formula | C19H15D6N3S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1216608-24-0 |
| Synonyms | |
| SMILES | [2H]C([2H])([2H])N(C([2H])([2H])[2H])CC(C)CN1C2=CC(C#N)=CC=C2SC3=CC=CC=C31 |
Biological Activity
| Description | Cyamemazine-d6 is a deuterated derivative of Cyamemazine, a neuroleptic agent characterized by its phenothiazine structure. This compound functions primarily as a potent antagonist of the 5-HT3 (Ki of 12 nM), 5-HT2A (Ki of 1.5 nM), and 5-HT2C (Ki of 75 nM) receptors, exhibiting notable anxiolytic and antipsychotic properties. Cyamemazine-d6 serves as a valuable stable isotope for studies involving pharmacokinetics, trace labeling, and metabolic research in the context of psychiatric disorders. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
