Product Data Sheet
GT-2016
Catalog No. A33953
GT-2016 is a potent and selective antagonist of the histamine H3 receptor, exhibiting a Ki value of 43.8 nM. This compound demonstrates high selectivity for the H3 receptor over H1 and H2 receptors and is inactive against histamine methyltransferase. GT-2016 is valuable for research into neurological disorders and sleep regulation, providing insights into histaminergic signaling pathways.
Chemical Information
| Catalog Num | A33953 |
|---|---|
| M. Wt | 317.47 |
| Formula | C19H31N3O |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 152241-24-2 |
| Synonyms | |
| SMILES | O=C(N1CCC(C2=CNC=N2)CC1)CCCCC3CCCCC3 |
Biological Activity
| Description | GT-2016 is a potent and selective antagonist of the histamine H3 receptor, exhibiting a Ki value of 43.8 nM. This compound demonstrates high selectivity for the H3 receptor over H1 and H2 receptors and is inactive against histamine methyltransferase. GT-2016 is valuable for research into neurological disorders and sleep regulation, providing insights into histaminergic signaling pathways. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
