Product Data Sheet
Pitolisant-d6
Catalog No. A34210
Pitolisant-d6 is a deuterium-labeled derivative of Pitolisant, which acts as a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). This stable isotope-labeled compound is utilized in pharmacokinetic studies and metabolic research, allowing for in-depth analysis of drug metabolism and interaction with the H3 receptor. It is an essential tool for researchers investigating sleep disorders and cognitive function modulation.
Chemical Information
| Catalog Num | A34210 |
|---|---|
| M. Wt | 301.88 |
| Formula | C17H20D6ClNO |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2416991-77-8 |
| Synonyms | Tiprolisant-d6 |
| SMILES | [2H]C(N1CCCCC1)([2H])C([2H])([2H])C([2H])([2H])OCCCC2=CC=C(C=C2)Cl |
Biological Activity
| Description | Pitolisant-d6 is a deuterium-labeled derivative of Pitolisant, which acts as a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). This stable isotope-labeled compound is utilized in pharmacokinetic studies and metabolic research, allowing for in-depth analysis of drug metabolism and interaction with the H3 receptor. It is an essential tool for researchers investigating sleep disorders and cognitive function modulation. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
