Product Data Sheet
PBRM1-BD2-IN-6
Catalog No. A40420
PBRM1-BD2-IN-6 is a selective inhibitor of the PBRM1 bromodomain, exhibiting a potent IC50 value of 0.22 μM. This compound demonstrates significant antiproliferative activity and is valuable for investigating PBRM1-dependent cancer mechanisms. Its application in research may aid in the development of targeted therapies for cancers that rely on PBRM1 modulation.
Chemical Information
| Catalog Num | A40420 |
|---|---|
| M. Wt | 286.76 |
| Formula | C16H15ClN2O |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2819989-67-6 |
| Synonyms | |
| SMILES | O=C1NC(C2=CC=CC(C)=C2C)NC3=C1C(Cl)=CC=C3 |
Biological Activity
| Description | PBRM1-BD2-IN-6 is a selective inhibitor of the PBRM1 bromodomain, exhibiting a potent IC50 value of 0.22 μM. This compound demonstrates significant antiproliferative activity and is valuable for investigating PBRM1-dependent cancer mechanisms. Its application in research may aid in the development of targeted therapies for cancers that rely on PBRM1 modulation. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
