Product Data Sheet
CPI-203-PEG1-C3-O-COOH
Catalog No. A40462
CPI-203-PEG1-C3-O-COOH is a BRD4 ligand-linker conjugate, designed to facilitate the synthesis of PROTAC (proteolysis-targeting chimera) molecules, specifically the BRD4 degrader ARV-771. This compound serves as a crucial component in targeted protein degradation research, enabling the selective modulation of BRD4 protein levels and aiding in the understanding of its biological functions. Its application is significant in therapeutic development for diseases associated with dysregulated BRD4 activity.
Chemical Information
| Catalog Num | A40462 |
|---|---|
| M. Wt | 560.06 |
| Formula | C26H30ClN5O5S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1997304-12-7 |
| Synonyms | |
| SMILES | CC1=C(C)C(C(C2=CC=C(Cl)C=C2)=N[C@@H](CC(NCCOCCCOCC(O)=O)=O)C3=NN=C(C)N34)=C4S1 |
Biological Activity
| Description | CPI-203-PEG1-C3-O-COOH is a BRD4 ligand-linker conjugate, designed to facilitate the synthesis of PROTAC (proteolysis-targeting chimera) molecules, specifically the BRD4 degrader ARV-771. This compound serves as a crucial component in targeted protein degradation research, enabling the selective modulation of BRD4 protein levels and aiding in the understanding of its biological functions. Its application is significant in therapeutic development for diseases associated with dysregulated BRD4 activity. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
