Product Data Sheet
BRD4-BD1/2-IN-2
Catalog No. A40506
BRD4-BD1/2-IN-2 is a highly selective inhibitor targeting the BD2 domain of BRD4, demonstrating IC50 values of less than 0.5 nM for BRD4 BD2 and approximately 300 nM for BRD4 BD1. This compound exhibits significant biological activity in modulating BRD4-related pathways, making it a valuable tool for research in oncology and epigenetic regulation. Its potency and specificity support further exploration of BRD4 as a therapeutic target in various diseases.
Chemical Information
| Catalog Num | A40506 |
|---|---|
| M. Wt | 527.61 |
| Formula | C30H33N5O4 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2743464-27-7 |
| Synonyms | |
| SMILES | O=C(C1=CC(C(C2=CC3=NN(CC(C)(C)O)C=C3C=C2OC4=C(C)C=CC=C4C)=CN5C)=C(N1)C5=O)NCC |
Biological Activity
| Description | BRD4-BD1/2-IN-2 is a highly selective inhibitor targeting the BD2 domain of BRD4, demonstrating IC50 values of less than 0.5 nM for BRD4 BD2 and approximately 300 nM for BRD4 BD1. This compound exhibits significant biological activity in modulating BRD4-related pathways, making it a valuable tool for research in oncology and epigenetic regulation. Its potency and specificity support further exploration of BRD4 as a therapeutic target in various diseases. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
