Product Data Sheet
Y08175
Catalog No. A40569
Y08175 is a highly potent inhibitor of the CBP bromodomain, demonstrating significant inhibitory capacity with IC50 values of 37 nM and 178.15 nM in AlphaScreen and HTRF assays, respectively. This compound is valuable for investigating the role of CBP in oncogenic processes, particularly in the context of prostate cancer research. Its ability to selectively target the CBP bromodomain makes it a useful tool for studying bromodomain-mediated transcriptional regulation and associated pathways.
Chemical Information
| Catalog Num | A40569 |
|---|---|
| M. Wt | 450.42 |
| Formula | C23H19FN4O5 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2223014-57-9 |
| Synonyms | |
| SMILES | O=C(O)C1=CC(C2=CN(C)N=C2)=C(F)C(NC(C3=CN(C(C)=O)C4=C3C=C(OC)C=C4)=O)=C1 |
Biological Activity
| Description | Y08175 is a highly potent inhibitor of the CBP bromodomain, demonstrating significant inhibitory capacity with IC50 values of 37 nM and 178.15 nM in AlphaScreen and HTRF assays, respectively. This compound is valuable for investigating the role of CBP in oncogenic processes, particularly in the context of prostate cancer research. Its ability to selectively target the CBP bromodomain makes it a useful tool for studying bromodomain-mediated transcriptional regulation and associated pathways. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
