Product Data Sheet
BET bromodomain inhibitor 2
Catalog No. A40571
BET Bromodomain Inhibitor 2 selectively targets the bromodomains of BET proteins, exhibiting a potent inhibitory effect with an IC50 of 14.1 µM. This compound is critical for modulating gene expression linked to cancer and inflammation by disrupting the interaction between acetylated histones and BET proteins. It is applicable in various research contexts, including oncology and epigenetics studies, providing invaluable insights into therapeutic strategies targeting bromodomain-containing proteins.
Chemical Information
| Catalog Num | A40571 |
|---|---|
| M. Wt | 446.56 |
| Formula | C23H30N2O5S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2414195-69-8 |
| Synonyms | |
| SMILES | CCN(S(=O)(C1=CC=C(C(C2=CC(OC)=C(C=C2)OC)=C1)[C@H]3CC(N(C3)C)=O)=O)CC |
Biological Activity
| Description | BET Bromodomain Inhibitor 2 selectively targets the bromodomains of BET proteins, exhibiting a potent inhibitory effect with an IC50 of 14.1 µM. This compound is critical for modulating gene expression linked to cancer and inflammation by disrupting the interaction between acetylated histones and BET proteins. It is applicable in various research contexts, including oncology and epigenetics studies, providing invaluable insights into therapeutic strategies targeting bromodomain-containing proteins. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
