Product Data Sheet
BRD4 Inhibitor-19
Catalog No. A40605
BRD4 Inhibitor-19 is a small molecule inhibitor targeting the bromodomain and extraterminal (BET) family, specifically inhibiting BRD4 with an IC50 of 55 nM at the BRD4-BD1 site. This compound exhibits significant anti-proliferative effects, making it a valuable tool in the study of multiple myeloma and related hematological malignancies. Researchers can utilize BRD4 Inhibitor-19 to explore the roles of BET proteins in cancer biology and evaluate potential therapeutic strategies in targeting aberrant gene expression.
Chemical Information
| Catalog Num | A40605 |
|---|---|
| M. Wt | 491.54 |
| Formula | C29H25N5O3 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2757865-63-5 |
| Synonyms | |
| SMILES | CC1=NOC(C)=C1C2=CC=C3C(C(N(C(N3C)=O)CC4=NN=C(O4)C5=CC=CC=C5)C6=CC=CC=C6)=C2 |
Biological Activity
| Description | BRD4 Inhibitor-19 is a small molecule inhibitor targeting the bromodomain and extraterminal (BET) family, specifically inhibiting BRD4 with an IC50 of 55 nM at the BRD4-BD1 site. This compound exhibits significant anti-proliferative effects, making it a valuable tool in the study of multiple myeloma and related hematological malignancies. Researchers can utilize BRD4 Inhibitor-19 to explore the roles of BET proteins in cancer biology and evaluate potential therapeutic strategies in targeting aberrant gene expression. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
